AZ1366 [Ligand Id: 10676] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| poly(ADP-ribose) polymerase 1 in Human [GtoPdb: 2771] [UniProtKB: P09874] | ||||||||
| GtoPdb | - | - | 6.25 | pIC50 | 559 | nM | IC50 | ACS Med Chem Lett (2015) 6: 254-9 [PMID:25815142] |
| poly(ADP-ribose) polymerase 2 in Human [GtoPdb: 2772] [UniProtKB: Q9UGN5] | ||||||||
| GtoPdb | - | - | 6.63 | pIC50 | 232 | nM | IC50 | ACS Med Chem Lett (2015) 6: 254-9 [PMID:25815142] |
| tankyrase in Human [GtoPdb: 3108] [UniProtKB: O95271] | ||||||||
| GtoPdb | - | - | 8.15 | pIC50 | 7 | nM | IC50 | ACS Med Chem Lett (2015) 6: 254-9 [PMID:25815142] |
| tankyrase 2 in Human [GtoPdb: 3109] [UniProtKB: Q9H2K2] | ||||||||
| GtoPdb | - | - | 8 | pIC50 | 10 | nM | IC50 | ACS Med Chem Lett (2015) 6: 254-9 [PMID:25815142] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
