golidocitinib [Ligand Id: 10744] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Janus kinase 1 in Human [GtoPdb: 2047] [UniProtKB: P23458] | ||||||||
| GtoPdb | Inhbition of JAK1 enzymatic activity. | - | 7.15 | pIC50 | 70 | nM | IC50 | J Med Chem (2020) 63: 4517-4527 [PMID:32297743] |
| Janus kinase 2 in Human [GtoPdb: 2048] [UniProtKB: O60674] | ||||||||
| GtoPdb | Inhbition of JAK2 enzymatic activity. | - | 4.82 | pIC50 | >15000 | nM | IC50 | J Med Chem (2020) 63: 4517-4527 [PMID:32297743] |
| tyrosine kinase 2 in Human [GtoPdb: 2269] [UniProtKB: P29597] | ||||||||
| GtoPdb | Inhbition of TYK2 enzymatic activity. | - | 5.55 | pIC50 | 2800 | nM | IC50 | J Med Chem (2020) 63: 4517-4527 [PMID:32297743] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
