[125I]CGP 64213 [Ligand Id: 1076] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1628547
  • GABAB1 in Rat [GtoPdb: 240] [UniProtKB: Q9Z0U4]
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  • GABAB receptor in Rat [GtoPdb: 242]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
GABAB1 in Rat [GtoPdb: 240] [UniProtKB: Q9Z0U4]
GtoPdb - - 8.9 pKd - - - Nature (1997) 386: 239-46 [PMID:9069281]
GABAB receptor in Rat [GtoPdb: 242]
GtoPdb - - 9 pKd 1 nM Kd Mol. Pharmacol. (2000) 57: 419-26 [PMID:10692480]

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]