ghrelin [Ligand Id: 1099] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| ghrelin receptor in Human [GtoPdb: 246] [UniProtKB: Q92847] | ||||||||
| GtoPdb | - | - | 9.44 | pKd | 0.36 | nM | Kd |
Mol Endocrinol (2003) 17: 2201-10 [PMID:12907757]; Mol Endocrinol (2005) 19: 2400-11 [PMID:15905359] |
| GtoPdb | - | - | 8.1 | pKi | - | - | - | J Endocrinol Invest (2001) 24: RC7-9 [PMID:11314756] |
| GtoPdb | - | - | 7.49 | pEC50 | 32 | nM | EC50 |
Mol Endocrinol (2005) 19: 2400-11 [PMID:15905359]; Mol Endocrinol (2000) 14: 160-9 [PMID:10628755] |
| GtoPdb | Measuring ghrelin-induced GHSR activation detected by β-arrestin recruitment in cells stably expressing hGHSR. | - | 8.15 | pEC50 | 7.1 | nM | EC50 | Cell Metab (2018) 27: 461-469.e6 [PMID:29233536] |
| GtoPdb | - | - | 9.47 | pEC50 | 0.34 | nM | EC50 |
Mol Endocrinol (2003) 17: 2201-10 [PMID:12907757]; J Biol Chem (2011) 286: 20845-60 [PMID:21402696] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
