BMS-986235 [Ligand Id: 11024] activity data from GtoPdb

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  • FPR1 in Human [GtoPdb: 222] [UniProtKB: P21462]
  • FPR1 in Mouse [GtoPdb: 222] [UniProtKB: P33766]
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  • FPR2/ALX in Human [GtoPdb: 223] [UniProtKB: P25090]
  • FPR2/ALX in Mouse [GtoPdb: 223] [UniProtKB: O88536]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
FPR1 in Human [GtoPdb: 222] [UniProtKB: P21462]
GtoPdb - - 6.4 pEC50 400 nM EC50 J. Med. Chem. (2020) null: null [PMID:32407089]
FPR1 in Mouse [GtoPdb: 222] [UniProtKB: P33766]
GtoPdb - - 6.3 pEC50 500 nM EC50 J. Med. Chem. (2020) null: null [PMID:32407089]
FPR2/ALX in Human [GtoPdb: 223] [UniProtKB: P25090]
GtoPdb - - 8.3 pEC50 5 nM EC50 J. Med. Chem. (2020) null: null [PMID:32407089]
FPR2/ALX in Mouse [GtoPdb: 223] [UniProtKB: O88536]
GtoPdb - - 9.3 pEC50 0.5 nM EC50 J. Med. Chem. (2020) null: null [PMID:32407089]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.