HTH-02-006 [Ligand Id: 11085] activity data from GtoPdb

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  • NUAK family kinase 1 in Human [GtoPdb: 2129] [UniProtKB: O60285]
  • This target only has 0 pki data point
  • 0
1 _lig_chart_1 NUAK family kinase 1 Human
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  • NUAK family, SNF1-like kinase, 2 in Human [GtoPdb: 2130] [UniProtKB: Q9H093]
  • This target only has 0 pki data point
  • 0
2 _lig_chart_2 NUAK family, SNF1-like kinase, 2 Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
NUAK family kinase 1 in Human [GtoPdb: 2129] [UniProtKB: O60285]
GtoPdb Determined in a radioactive (33P-ATP) filter-binding assay. - 8.1 pIC50 8 nM IC50 Nat Commun (2018) 9: 4834 [PMID:30446657]
NUAK family, SNF1-like kinase, 2 in Human [GtoPdb: 2130] [UniProtKB: Q9H093]
GtoPdb Determined in a radioactive (33P-ATP) filter-binding assay. - 6.9 pIC50 126 nM IC50 Nat Commun (2018) 9: 4834 [PMID:30446657]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.