martinostat [Ligand Id: 11118] activity data from GtoPdb

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  • histone deacetylase 2 in Human [GtoPdb: 2616] [UniProtKB: Q92769]
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  • histone deacetylase 3 in Human [GtoPdb: 2617] [UniProtKB: O15379]
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  • histone deacetylase 6 in Human [GtoPdb: 2618] [UniProtKB: Q9UBN7]
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  • histone deacetylase 1 in Human [GtoPdb: 2658] [UniProtKB: Q13547]
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  • histone deacetylase 4 in Human [GtoPdb: 2659] [UniProtKB: P56524]
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  • histone deacetylase 5 in Human [GtoPdb: 2660] [UniProtKB: Q9UQL6]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
histone deacetylase 2 in Human [GtoPdb: 2616] [UniProtKB: Q92769]
GtoPdb - - 8.7 pIC50 2 nM IC50 J Med Chem (2014) 57: 7999-8009 [PMID:25203558]
histone deacetylase 3 in Human [GtoPdb: 2617] [UniProtKB: O15379]
GtoPdb - - 9.22 pIC50 0.6 nM IC50 J Med Chem (2014) 57: 7999-8009 [PMID:25203558]
histone deacetylase 6 in Human [GtoPdb: 2618] [UniProtKB: Q9UBN7]
GtoPdb - - 8.39 pIC50 4.1 nM IC50 J Med Chem (2014) 57: 7999-8009 [PMID:25203558]
histone deacetylase 1 in Human [GtoPdb: 2658] [UniProtKB: Q13547]
GtoPdb - - 9.52 pIC50 0.3 nM IC50 J Med Chem (2014) 57: 7999-8009 [PMID:25203558]
histone deacetylase 4 in Human [GtoPdb: 2659] [UniProtKB: P56524]
GtoPdb - - 5.71 pIC50 1970 nM IC50 J Med Chem (2014) 57: 7999-8009 [PMID:25203558]
histone deacetylase 5 in Human [GtoPdb: 2660] [UniProtKB: Q9UQL6]
GtoPdb - - 6.45 pIC50 352 nM IC50 J Med Chem (2014) 57: 7999-8009 [PMID:25203558]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.