suprastat [Ligand Id: 11220] activity data from GtoPdb

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  • histone deacetylase 2 in Human [GtoPdb: 2616] [UniProtKB: Q92769]
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  • histone deacetylase 3 in Human [GtoPdb: 2617] [UniProtKB: O15379]
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  • histone deacetylase 6 in Human [GtoPdb: 2618] [UniProtKB: Q9UBN7]
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  • histone deacetylase 8 in Human [GtoPdb: 2619] [UniProtKB: Q9BY41]
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  • histone deacetylase 1 in Human [GtoPdb: 2658] [UniProtKB: Q13547]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
histone deacetylase 2 in Human [GtoPdb: 2616] [UniProtKB: Q92769]
GtoPdb - - 6.75 pIC50 176 nM IC50 J Med Chem (2020) 63: 10246-10262 [PMID:32815366]
histone deacetylase 3 in Human [GtoPdb: 2617] [UniProtKB: O15379]
GtoPdb - - 6.45 pIC50 352 nM IC50 J Med Chem (2020) 63: 10246-10262 [PMID:32815366]
histone deacetylase 6 in Human [GtoPdb: 2618] [UniProtKB: Q9UBN7]
GtoPdb - - 9.4 pIC50 0.4 nM IC50 J Med Chem (2020) 63: 10246-10262 [PMID:32815366]
histone deacetylase 8 in Human [GtoPdb: 2619] [UniProtKB: Q9BY41]
GtoPdb - - 6.3 pIC50 498 nM IC50 J Med Chem (2020) 63: 10246-10262 [PMID:32815366]
histone deacetylase 1 in Human [GtoPdb: 2658] [UniProtKB: Q13547]
GtoPdb - - 6.93 pIC50 117 nM IC50 J Med Chem (2020) 63: 10246-10262 [PMID:32815366]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.