edaxeterkib [Ligand Id: 11411] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • mitogen-activated protein kinase 1 in Human [GtoPdb: 1495] [UniProtKB: P28482]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
mitogen-activated protein kinase 1 in Human [GtoPdb: 1495] [UniProtKB: P28482]
GtoPdb Binned IC50 value from patent; determined using the proprietary Z'- LYTE kinase assay. - 7.3 pIC50 <50 nM IC50 WO2015051341A1. Inhibitors of erk and methods of use (2015)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.