CC-90005 [Ligand Id: 11659] activity data from GtoPdb

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  • protein kinase C delta in Human [GtoPdb: 1485] [UniProtKB: Q05655]
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  • protein kinase C theta in Human [GtoPdb: 1488] [UniProtKB: Q04759]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
protein kinase C delta in Human [GtoPdb: 1485] [UniProtKB: Q05655]
GtoPdb - - 5.35 pIC50 4440 nM IC50 J Med Chem (2021) 64: 11886-11903 [PMID:34355886]
protein kinase C theta in Human [GtoPdb: 1488] [UniProtKB: Q04759]
GtoPdb - - 8.1 pIC50 8 nM IC50 J Med Chem (2021) 64: 11886-11903 [PMID:34355886]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.