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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| epidermal growth factor receptor in Human [GtoPdb: 1797] [UniProtKB: P00533] | ||||||||
| GtoPdb | Inhibition of WT EGFR phosphorylation in A431 cells | - | 7.09 | pIC50 | 80.4 | nM | IC50 | WO2019149164A1. Erbb/btk inhibitors (2019) |
| Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187] | ||||||||
| GtoPdb | Inhibition of BTK phosphorylation in Ramos cells (B lymphocyte cell line) | - | 8.54 | pIC50 | 2.9 | nM | IC50 | WO2019149164A1. Erbb/btk inhibitors (2019) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.