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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| ATM serine/threonine kinase in Human [GtoPdb: 1934] [UniProtKB: Q13315] | ||||||||
| GtoPdb | - | - | 4.71 | pIC50 | 19300 | nM | IC50 | J Med Chem (2021) 64: 12723-12737 [PMID:34428039] |
| ATR checkpoint kinase in Human [GtoPdb: 1935] [UniProtKB: Q13535] | ||||||||
| GtoPdb | - | - | 6.4 | pIC50 | 394 | nM | IC50 | J Med Chem (2021) 64: 12723-12737 [PMID:34428039] |
| phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit beta in Human [GtoPdb: 2154] [UniProtKB: P42338] | ||||||||
| GtoPdb | - | - | 6.93 | pIC50 | 117 | nM | IC50 | J Med Chem (2021) 64: 12723-12737 [PMID:34428039] |
| protein kinase, DNA-activated, catalytic subunit in Human [GtoPdb: 2800] [UniProtKB: P78527] | ||||||||
| GtoPdb | - | - | 7.09 | pIC50 | 81 | nM | IC50 | J Med Chem (2021) 64: 12723-12737 [PMID:34428039] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.