XR8-24 [Ligand Id: 11766] activity data from GtoPdb

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  • CoV Papain-like protease in SARS-CoV-2 [GtoPdb: 3132] [UniProtKB: P0DTC1]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CoV Papain-like protease in SARS-CoV-2 [GtoPdb: 3132] [UniProtKB: P0DTC1]
GtoPdb - - 6.43 pKd 372 nM Kd J Med Chem (2022) 65: 2940-2955 [PMID:34665619]
GtoPdb - - 6.41 pIC50 390 nM IC50 J Med Chem (2022) 65: 2940-2955 [PMID:34665619]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.