zilurgisertib [Ligand Id: 11888] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| activin A receptor type IL in Human [GtoPdb: 1784] [UniProtKB: P37023] | ||||||||
| GtoPdb | - | - | 6.49 | pIC50 | 323 | nM | IC50 | US20210155606A1. Aminopyridine derivatives and their use as selective alk-2 inhibitors (2021) |
| activin A receptor type 1 in Human [GtoPdb: 1785] [UniProtKB: Q04771] | ||||||||
| GtoPdb | - | - | 7.64 | pIC50 | 23 | nM | IC50 | US20210155606A1. Aminopyridine derivatives and their use as selective alk-2 inhibitors (2021) |
| bone morphogenetic protein receptor type IA in Human [GtoPdb: 1786] [UniProtKB: P36894] | ||||||||
| GtoPdb | - | - | 6.04 | pIC50 | 914 | nM | IC50 | US20210155606A1. Aminopyridine derivatives and their use as selective alk-2 inhibitors (2021) |
| transforming growth factor beta receptor 1 in Human [GtoPdb: 1788] [UniProtKB: P36897] | ||||||||
| GtoPdb | - | - | 5.2 | pIC50 | 6280 | nM | IC50 | US20210155606A1. Aminopyridine derivatives and their use as selective alk-2 inhibitors (2021) |
| bone morphogenetic protein receptor type IB in Human [GtoPdb: 1789] [UniProtKB: O00238] | ||||||||
| GtoPdb | - | - | 5.48 | pIC50 | 3300 | nM | IC50 | US20210155606A1. Aminopyridine derivatives and their use as selective alk-2 inhibitors (2021) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
