compound 14 [PMID: 34333981] [Ligand Id: 11896] activity data from GtoPdb

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  • microtubule affinity regulating kinase 3 in Human [GtoPdb: 2099] [UniProtKB: P27448]
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  • microtubule affinity regulating kinase 4 in Human [GtoPdb: 2100] [UniProtKB: Q96L34]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
microtubule affinity regulating kinase 3 in Human [GtoPdb: 2099] [UniProtKB: P27448]
GtoPdb - - 5.4 pIC50 4015 nM IC50 J Med Chem (2022) 65: 1313-1328 [PMID:34333981]
microtubule affinity regulating kinase 4 in Human [GtoPdb: 2100] [UniProtKB: Q96L34]
GtoPdb - - 6.09 pIC50 808 nM IC50 J Med Chem (2022) 65: 1313-1328 [PMID:34333981]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.