SAGE-718 [Ligand Id: 12050] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| GluN2A in Human [GtoPdb: 456] [UniProtKB: Q12879] | ||||||||
| GtoPdb | Value obtained using automated patch clamp electrophysiology in HEK293 cells stably expressing recombinant human GluN1/GluN2A Rs | - | 7.07 | pEC50 | 86 | nM | EC50 | J Med Chem (2022) 65: 9063-9075 [PMID:35785990] |
| GluN2B in Human [GtoPdb: 457] [UniProtKB: Q13224] | ||||||||
| GtoPdb | Value obtained using automated patch clamp electrophysiology in HEK293 cells stably expressing recombinant human GluN1/GluN2B Rs | - | 7.1 | pEC50 | 79 | nM | EC50 | J Med Chem (2022) 65: 9063-9075 [PMID:35785990] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
