Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
fibroblast growth factor receptor 1 in Human [GtoPdb: 1808] [UniProtKB: P11362] | ||||||||
GtoPdb | - | - | 7.68 | pIC50 | 21 | nM | IC50 | J Med Chem (2022) 65: 15433-15442 [PMID:36356320] |
fibroblast growth factor receptor 2 in Human [GtoPdb: 1809] [UniProtKB: P21802] | ||||||||
GtoPdb | - | - | 9 | pIC50 | 1 | nM | IC50 | J Med Chem (2022) 65: 15433-15442 [PMID:36356320] |
fibroblast growth factor receptor 3 in Human [GtoPdb: 1810] [UniProtKB: P22607] | ||||||||
GtoPdb | Inhibition of FGFR3V555L in vitro. | - | 8.57 | pIC50 | 2.7 | nM | IC50 | J Med Chem (2022) 65: 15433-15442 [PMID:36356320] |
GtoPdb | Inhibition of WT FGFR3 in vitro. | - | 9.3 | pIC50 | 0.5 | nM | IC50 | J Med Chem (2022) 65: 15433-15442 [PMID:36356320] |
fibroblast growth factor receptor 4 in Human [GtoPdb: 1811] [UniProtKB: P22455] | ||||||||
GtoPdb | - | - | 6.84 | pIC50 | 145 | nM | IC50 | J Med Chem (2022) 65: 15433-15442 [PMID:36356320] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.