lartesertib [Ligand Id: 12319] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| ATM serine/threonine kinase in Human [GtoPdb: 1934] [UniProtKB: Q13315] | ||||||||
| GtoPdb | Inhibition in a biochemical assay, ATP at 10 μM | - | 9.7 | pIC50 | 0.2 | nM | IC50 | WO2020193660A1. Imidazolonylquinoline compounds and therapeutic uses thereof (2020) |
| protein kinase, DNA-activated, catalytic subunit in Human [GtoPdb: 2800] [UniProtKB: P78527] | ||||||||
| GtoPdb | - | - | 6.22 | pIC50 | 600 | nM | IC50 | WO2020193660A1. Imidazolonylquinoline compounds and therapeutic uses thereof (2020) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
