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ChEMBL ligand: CHEMBL512 |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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H2 receptor in Human [GtoPdb: 263] [UniProtKB: P25021] | ||||||||
GtoPdb | - | - | 7.1 | pKi | 79.4 | nM | Ki | Br. J. Pharmacol. (1994) 112: 847-54 [PMID:7921611] |
H2 receptor in Rat [GtoPdb: 263] [UniProtKB: P25102] | ||||||||
GtoPdb | - | - | 6.2 | pKi | 631 | nM | Ki | Br. J. Pharmacol. (1997) 122: 867-74 [PMID:9384502] |
ChEMBL data shown on this page come from version 27:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]