resencatinib [Ligand Id: 12381] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| kinase insert domain receptor in Human [GtoPdb: 1813] [UniProtKB: P35968] | ||||||||
| GtoPdb | - | - | 7.66 | pIC50 | 21.7 | nM | IC50 | WO2020228756A1. Inhibitor containing bicyclic derivative, preparation method therefor and use thereof (2020) |
| ret proto-oncogene in Human [GtoPdb: 2185] [UniProtKB: P07949] | ||||||||
| GtoPdb | Inhibitory potency vs. WT hRET | - | 9.47 | pIC50 | 0.34 | nM | IC50 | WO2020228756A1. Inhibitor containing bicyclic derivative, preparation method therefor and use thereof (2020) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
