[3H]GR 125,743 [Ligand Id: 131] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1628631
  • 5-HT1B receptor in Human [GtoPdb: 2] [UniProtKB: P28222]
  • This target only has 0 pki data point
1 CHEMBL1628631_lig_chart_1 5-HT1B receptor Human
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  • 5-HT1D receptor in Human [GtoPdb: 3] [UniProtKB: P28221]
  • This target only has 0 pki data point
2 CHEMBL1628631_lig_chart_2 5-HT1D receptor Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
5-HT1B receptor in Human [GtoPdb: 2] [UniProtKB: P28222]
GtoPdb - - 9.2 pKd 0.71 nM Kd Eur. J. Pharmacol. (1999) 380: 171-81 [PMID:10513577];
FEBS Lett. (1999) 456: 63-7 [PMID:10452531]
5-HT1D receptor in Human [GtoPdb: 3] [UniProtKB: P28221]
GtoPdb - - 8.6 pKd 2.8 nM Kd FEBS Lett. (1999) 456: 63-7 [PMID:10452531]

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]