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1
_lig_chart_1
MC1 receptor
Human
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2
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MC3 receptor
Human
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3
_lig_chart_3
MC4 receptor
Human
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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MC1 receptor in Human [GtoPdb: 282] [UniProtKB: Q01726] | ||||||||
GtoPdb | - | - | 7 | pKd | - | - | - | Neuropeptides (1999) 33: 191-6 [PMID:10657491] |
MC3 receptor in Human [GtoPdb: 284] [UniProtKB: P41968] | ||||||||
GtoPdb | - | - | 7.3 | pKd | - | - | - | Neuropeptides (1999) 33: 191-6 [PMID:10657491] |
MC4 receptor in Human [GtoPdb: 285] [UniProtKB: P32245] | ||||||||
GtoPdb | - | - | 8.5 | pKd | 3.16 | nM | Kd | Br. J. Pharmacol. (1999) 126: 27-34 [PMID:10051117] |
GtoPdb | - | - | 8.5 | pKi | 3.2 | nM | Ki | Br. J. Pharmacol. (1998) 124: 75-82 [PMID:9630346] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.