HS014 [Ligand Id: 1321] activity data from GtoPdb

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  • MC1 receptor in Human [GtoPdb: 282] [UniProtKB: Q01726]
  • This target only has 0 pki data point
1 _lig_chart_1 MC1 receptor Human
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  • MC3 receptor in Human [GtoPdb: 284] [UniProtKB: P41968]
  • This target only has 0 pki data point
2 _lig_chart_2 MC3 receptor Human
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  • MC4 receptor in Human [GtoPdb: 285] [UniProtKB: P32245]
  • This target only has 1 pki data point
3 _lig_chart_3 MC4 receptor Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
MC1 receptor in Human [GtoPdb: 282] [UniProtKB: Q01726]
GtoPdb - - 7 pKd - - - Neuropeptides (1999) 33: 191-6 [PMID:10657491]
MC3 receptor in Human [GtoPdb: 284] [UniProtKB: P41968]
GtoPdb - - 7.3 pKd - - - Neuropeptides (1999) 33: 191-6 [PMID:10657491]
MC4 receptor in Human [GtoPdb: 285] [UniProtKB: P32245]
GtoPdb - - 8.5 pKd 3.16 nM Kd Br. J. Pharmacol. (1999) 126: 27-34 [PMID:10051117]
GtoPdb - - 8.5 pKi 3.2 nM Ki Br. J. Pharmacol. (1998) 124: 75-82 [PMID:9630346]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.