PG-901 [Ligand Id: 1341] activity data from GtoPdb

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  • MC3 receptor in Human [GtoPdb: 284] [UniProtKB: P41968]
  • This target only has 0 pki data point
1 _lig_chart_1 MC3 receptor Human
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  • MC4 receptor in Human [GtoPdb: 285] [UniProtKB: P32245]
  • This target only has 0 pki data point
2 _lig_chart_2 MC4 receptor Human
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  • MC5 receptor in Human [GtoPdb: 286] [UniProtKB: P33032]
  • This target only has 0 pki data point
3 _lig_chart_3 MC5 receptor Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
MC3 receptor in Human [GtoPdb: 284] [UniProtKB: P41968]
GtoPdb - - 9.7 pIC50 - - - J. Med. Chem. (2002) 45: 5287-94 [PMID:12431055]
MC4 receptor in Human [GtoPdb: 285] [UniProtKB: P32245]
GtoPdb - - 8.1 pIC50 - - - J. Med. Chem. (2002) 45: 5287-94 [PMID:12431055]
MC5 receptor in Human [GtoPdb: 286] [UniProtKB: P33032]
GtoPdb - - 10.5 pIC50 - - - J. Med. Chem. (2002) 45: 5287-94 [PMID:12431055]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.