A-910 [Ligand Id: 13579] activity data from GtoPdb

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  • AXL receptor tyrosine kinase in Human [GtoPdb: 1835] [UniProtKB: P30530]
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  • TYRO3 protein tyrosine kinase in Human [GtoPdb: 1836] [UniProtKB: Q06418]
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  • MER proto-oncogene, tyrosine kinase in Human [GtoPdb: 1837] [UniProtKB: Q12866]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
AXL receptor tyrosine kinase in Human [GtoPdb: 1835] [UniProtKB: P30530]
GtoPdb - - 8.09 pIC50 8.2 nM IC50 J Med Chem (2024) 67: 17000-17032 [PMID:39283694]
TYRO3 protein tyrosine kinase in Human [GtoPdb: 1836] [UniProtKB: Q06418]
GtoPdb - - 6.26 pIC50 555 nM IC50 J Med Chem (2024) 67: 17000-17032 [PMID:39283694]
MER proto-oncogene, tyrosine kinase in Human [GtoPdb: 1837] [UniProtKB: Q12866]
GtoPdb Inhibition of Mer TK in Ba/F3 cells - 8.38 pIC50 4.2 nM IC50 J Med Chem (2024) 67: 17000-17032 [PMID:39283694]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.