Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
ChEMBL ligand: CHEMBL3143516 |
---|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
Motilin receptor in Rabbit (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5306] [UniProtKB: A5A4K8] | ||||||||
ChEMBL | Inhibition of the motilin receptor (MTL-R) | B | 8 | pIC50 | 10 | nM | IC50 | J Med Chem (2002) 45: 670-675 [PMID:11806718] |
motilin receptor in Rabbit [GtoPdb: 297] | ||||||||
GtoPdb | - | - | 8 | pIC50 | - | - | - | J Med Chem (2002) 45: 670-5 [PMID:11806718] |
GtoPdb | - | - | 7.5 | pA2 | - | - | - |
Clin Exp Pharmacol Physiol (1999) 26: 242-5 [PMID:10081621]; J Pharmacol Exp Ther (1995) 273: 624-8 [PMID:7752063] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]