GM-109 [Ligand Id: 1466] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL3143516
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  • motilin receptor in Rabbit [GtoPdb: 297]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Motilin receptor in Rabbit (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5306] [UniProtKB: A5A4K8]
ChEMBL Inhibition of the motilin receptor (MTL-R) B 8 pIC50 10 nM IC50 J. Med. Chem. (2002) 45: 670-675 [PMID:11806718]
motilin receptor in Rabbit [GtoPdb: 297]
GtoPdb - - 8 pIC50 - - - J Med Chem (2002) 45: 670-5 [PMID:11806718]
GtoPdb - - 7.5 pA2 - - - Clin Exp Pharmacol Physiol (1999) 26: 242-5 [PMID:10081621];
J Pharmacol Exp Ther (1995) 273: 624-8 [PMID:7752063]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]