[Leu]enkephalin [Ligand Id: 1613] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL15038
  • δ receptor in Human [GtoPdb: 317] [UniProtKB: P41143]
  • δ receptor in Mouse [GtoPdb: 317] [UniProtKB: P32300]
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  • κ receptor in Rat [GtoPdb: 318] [UniProtKB: P34975]
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  • μ receptor in Human [GtoPdb: 319] [UniProtKB: P35372]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
δ receptor in Human [GtoPdb: 317] [UniProtKB: P41143]
GtoPdb - - 8.7 pKi - - - NIDA Res Monogr (1998) 178: 440-66 [PMID:9686407]
δ receptor in Mouse [GtoPdb: 317] [UniProtKB: P32300]
GtoPdb - - 8.4 pKi - - - Mol Pharmacol (1994) 45: 330-4 [PMID:8114680]
κ receptor in Rat [GtoPdb: 318] [UniProtKB: P34975]
GtoPdb - - 6 pKi - - - Proc Natl Acad Sci USA (1993) 90: 9954-8 [PMID:8234341]
μ receptor in Human [GtoPdb: 319] [UniProtKB: P35372]
GtoPdb - - 8.1 pKi - - - NIDA Res Monogr (1998) 178: 440-66 [PMID:9686407]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]