Org 12962 [Ligand Id: 170] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL506999
  • 5-HT2A receptor in Human [GtoPdb: 6] [UniProtKB: P28223]
  • This target only has 1 pki data point
1 CHEMBL506999_lig_chart_1 5-HT2A receptor Human
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  • 5-HT2B receptor in Human [GtoPdb: 7] [UniProtKB: P41595]
  • This target only has 1 pki data point
2 CHEMBL506999_lig_chart_2 5-HT2B receptor Human
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  • 5-HT2C receptor in Human [GtoPdb: 8] [UniProtKB: P28335]
  • This target only has 1 pki data point
3 CHEMBL506999_lig_chart_3 5-HT2C receptor Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
5-HT2A receptor in Human [GtoPdb: 6] [UniProtKB: P28223]
GtoPdb - - 7.5 pKi - - - Naunyn Schmiedebergs Arch. Pharmacol. (2004) 370: 114-23 [PMID:15322733]
5-HT2B receptor in Human [GtoPdb: 7] [UniProtKB: P41595]
GtoPdb - - 7 pKi - - - Naunyn Schmiedebergs Arch. Pharmacol. (2004) 370: 114-23 [PMID:15322733]
5-HT2C receptor in Human [GtoPdb: 8] [UniProtKB: P28335]
GtoPdb - - 7.8 pKi - - - Naunyn Schmiedebergs Arch. Pharmacol. (2004) 370: 114-23 [PMID:15322733]

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]