L-644,698 [Ligand Id: 1879] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL117168
  • DP1 receptor in Human [GtoPdb: 338] [UniProtKB: Q13258]
  • DP1 receptor in Rat [GtoPdb: 338] [UniProtKB: Q9R261]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
DP1 receptor in Human [GtoPdb: 338] [UniProtKB: Q13258]
GtoPdb - - 9.3 pKi - - - Eur. J. Pharmacol. (1999) 377: 101-15 [PMID:10448933];
Br. J. Pharmacol. (1998) 123: 1317-24 [PMID:9579725]
DP1 receptor in Rat [GtoPdb: 338] [UniProtKB: Q9R261]
GtoPdb - - 6.8 pKi - - - Eur. J. Pharmacol. (1999) 377: 101-15 [PMID:10448933]

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]