ChEMBL ligand: CHEMBL264421
TP receptor/Thromboxane A2 receptor in Human [ChEMBL: CHEMBL2069] [GtoPdb: 346] [UniProtKB: P21731] There should be some charts here, you may need to enable JavaScript!
DP1 receptor in Human [GtoPdb: 338] [UniProtKB: Q13258] There should be some charts here, you may need to enable JavaScript!
DP2 receptor in Human [GtoPdb: 339] [UniProtKB: Q9Y5Y4] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
TP receptor/Thromboxane A2 receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2069] [GtoPdb: 346] [UniProtKB: P21731]
ChEMBL	Binding affinity to human recombinant TP receptor by radioligand competition binding assay	B	7.77	pKi	17	nM	Ki	Bioorg Med Chem Lett (2008) 18: 2696-2700 [PMID:18359630]
DP1 receptor in Human [GtoPdb: 338] [UniProtKB: Q13258]
GtoPdb	-	-	7.4	pKi	-	-	-	Mol Pharmacol (2005) 67: 1834-9 [PMID:15755909]
DP2 receptor in Human [GtoPdb: 339] [UniProtKB: Q9Y5Y4]
GtoPdb	-	-	7.32	pKi	48	nM	Ki	Mol Pharmacol (2005) 67: 1834-9 [PMID:15755909]

ChEMBL data shown on this page come from version 33:

Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]