ONO-8713 [Ligand Id: 1921] activity data from GtoPdb

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  • EP1 receptor in Human [GtoPdb: 340] [UniProtKB: P34995]
  • EP1 receptor in Mouse [GtoPdb: 340] [UniProtKB: P35375]
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  • EP3 receptor in Mouse [GtoPdb: 342] [UniProtKB: P30557]
  • EP3 receptor in Rat [GtoPdb: 342] [UniProtKB: P34980]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
EP1 receptor in Human [GtoPdb: 340] [UniProtKB: P34995]
GtoPdb - - 8 pKi - - - Bioorg Med Chem Lett (1999) 9: 2699-704 [PMID:10509919]
EP1 receptor in Mouse [GtoPdb: 340] [UniProtKB: P35375]
GtoPdb - - 9.5 pKi - - - Cancer Lett (2000) 156: 57-61 [PMID:10840160]
EP3 receptor in Mouse [GtoPdb: 342] [UniProtKB: P30557]
GtoPdb - - 5 pKi >10000 nM Ki Cancer Lett (2000) 156: 57-61 [PMID:10840160]
EP3 receptor in Rat [GtoPdb: 342] [UniProtKB: P34980]
GtoPdb - - 8.49 pKi 3.2 nM Ki Eur J Pharmacol (1997) 340: 227-41 [PMID:9537820]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.