pasireotide [Ligand Id: 2018] activity data from GtoPdb

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  • SST1 receptor in Human [GtoPdb: 355] [UniProtKB: P30872]
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  • SST2 receptor in Human [GtoPdb: 356] [UniProtKB: P30874]
  • SST2 receptor in Rat [GtoPdb: 356] [UniProtKB: P30680]
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  • SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
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  • SST5 receptor in Human [GtoPdb: 359] [UniProtKB: P35346]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
SST1 receptor in Human [GtoPdb: 355] [UniProtKB: P30872]
GtoPdb - - 8 pIC50 - - - Neuroendocrinology (2004) 80 Suppl 1: 47-50 [PMID:15477717]
SST2 receptor in Human [GtoPdb: 356] [UniProtKB: P30874]
GtoPdb - - 9 pIC50 - - - Neuroendocrinology (2004) 80 Suppl 1: 47-50 [PMID:15477717]
SST2 receptor in Rat [GtoPdb: 356] [UniProtKB: P30680]
GtoPdb - - 5 pEC50 >10000 nM EC50 Mol. Endocrinol. (2010) 24: 240-9 [PMID:19910453]
GtoPdb - - 7.63 pEC50 23.3 nM EC50 Mol. Endocrinol. (2011) 25: 1040-54 [PMID:21493671]
GtoPdb - - 9.07 pEC50 0.86 nM EC50 Mol. Endocrinol. (2010) 24: 240-9 [PMID:19910453];
Mol. Endocrinol. (2011) 25: 1040-54 [PMID:21493671]
SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
GtoPdb - - 8.8 pIC50 - - - Neuroendocrinology (2004) 80 Suppl 1: 47-50 [PMID:15477717]
SST5 receptor in Human [GtoPdb: 359] [UniProtKB: P35346]
GtoPdb - - 9.8 pIC50 - - - Neuroendocrinology (2004) 80 Suppl 1: 47-50 [PMID:15477717]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.