L-363,301 [Ligand Id: 2047] activity data from GtoPdb

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  • SST2 receptor in Human [GtoPdb: 356] [UniProtKB: P30874]
  • SST2 receptor in Mouse [GtoPdb: 356] [UniProtKB: P30875]
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  • SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
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  • SST5 receptor in Human [GtoPdb: 359] [UniProtKB: P35346]
  • SST5 receptor in Rat [GtoPdb: 359] [UniProtKB: P30938]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
SST2 receptor in Human [GtoPdb: 356] [UniProtKB: P30874]
GtoPdb - - 8.5 pKi - - - Naunyn Schmiedebergs Arch. Pharmacol. (1998) 357: 483-9 [PMID:9650799];
Naunyn Schmiedebergs Arch. Pharmacol. (1999) 360: 488-99 [PMID:10598788]
SST2 receptor in Mouse [GtoPdb: 356] [UniProtKB: P30875]
GtoPdb - - 9.1 pIC50 - - - Mol. Pharmacol. (1993) 43: 838-44 [PMID:8100350];
Metab. Clin. Exp. (1996) 45: 12-3 [PMID:8769370]
SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
GtoPdb - - 7 pKi - - - Naunyn Schmiedebergs Arch. Pharmacol. (1998) 357: 483-9 [PMID:9650799];
Naunyn Schmiedebergs Arch. Pharmacol. (1999) 360: 488-99 [PMID:10598788]
SST5 receptor in Human [GtoPdb: 359] [UniProtKB: P35346]
GtoPdb - - 9.5 pKi - - - Naunyn Schmiedebergs Arch. Pharmacol. (1998) 357: 483-9 [PMID:9650799];
Naunyn Schmiedebergs Arch. Pharmacol. (1999) 360: 488-99 [PMID:10598788]
SST5 receptor in Rat [GtoPdb: 359] [UniProtKB: P30938]
GtoPdb - - 8.3 pKd - - - Neuropharmacology (2000) 39: 1451-62 [PMID:10818261]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.