[Ac-His1]PACAP-27 [Ligand Id: 2263] activity data from GtoPdb

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  • PAC1 receptor in Rat [GtoPdb: 370] [UniProtKB: P32215]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
PAC1 receptor in Rat [GtoPdb: 370] [UniProtKB: P32215]
GtoPdb inhibition of [125I]-[Ac-His1]PACAP-27 binding to membranes from CHO cells stably expressing the rat PAC1 receptor isoform lacking the hip and hop exons - 8 pKi 10 nM Ki Eur. J. Pharmacol. (1995) 288: 259-67 [PMID:7774670]
GtoPdb inhibition of [125I]-[Ac-His1]PACAP-27 binding to membranes from CHO cells stably expressing the rat PAC1 receptor isoform including the hop1 exon - 8.3 pKi 5 nM Ki Eur. J. Pharmacol. (1995) 288: 259-67 [PMID:7774670]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.