N-stearyl-[Nle17] neurotensin-(6-11)/VIP-(7-28) [Ligand Id: 2266] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| PAC1 receptor in Human [GtoPdb: 370] [UniProtKB: P41586] | ||||||||
| GtoPdb | inhibition of [125I]-PACAP-27 binding to membranes from NIH/3T3 cells stably expressing the recombinant receptor | - | 7.2 | pIC50 | 65 | nM | IC50 | J Mol Neurosci (2002) 18: 29-35 [PMID:11931347] |
| VPAC1 receptor in Human [GtoPdb: 371] [UniProtKB: P32241] | ||||||||
| GtoPdb | inhibition of [125I]-VIP binding to membranes from CHO cells stably expressing the recombinant receptor | - | 7.5 | pIC50 | 30 | nM | IC50 | J Mol Neurosci (2002) 18: 29-35 [PMID:11931347] |
| VPAC2 receptor in Human [GtoPdb: 372] [UniProtKB: P41587] | ||||||||
| GtoPdb | inhibition of [125I]-VIP binding to membranes from CHO cells stably expressing the recombinant receptor | - | 7.3 | pIC50 | 50 | nM | IC50 | J Mol Neurosci (2002) 18: 29-35 [PMID:11931347] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
