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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference | 
|---|---|---|---|---|---|---|---|---|
| Kv1.1 in Human [GtoPdb: 538] [UniProtKB: Q09470] | ||||||||
| GtoPdb | - | - | 8.4 | pIC50 | 4.2 | nM | IC50 | Toxicon (2014) 87: 6-16 [PMID:24878374] | 
| Kv1.1 in Rat [GtoPdb: 538] [UniProtKB: P10499] | ||||||||
| GtoPdb | - | - | 8.3 | pIC50 | 5.46 | nM | IC50 | J Biol Chem (1997) 272: 27577-81 [PMID:9346893] | 
| Kv1.2 in Human [GtoPdb: 539] [UniProtKB: P16389] | ||||||||
| GtoPdb | - | - | 11.2 | pIC50 | 0.01 | nM | IC50 | Toxicon (2014) 87: 6-16 [PMID:24878374] | 
| Kv1.3 in Human [GtoPdb: 540] [UniProtKB: P22001] | ||||||||
| GtoPdb | - | - | 10.3 | pIC50 | 0.05 | nM | IC50 | J Biol Chem (2000) 275: 37137-49 [PMID:10961988]; J Biol Chem (1993) 268: 18866-74 [PMID:8360176] | 
| Kv1.7 in Mouse [GtoPdb: 544] [UniProtKB: Q17ST2] | ||||||||
| GtoPdb | - | - | 6.9 | pIC50 | - | - | - | J Biol Chem (1998) 273: 5851-7 [PMID:9488722] | 
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.