androstenol [Ligand Id: 2761] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL142348 (Androstenol)
  • Constitutive androstane receptor in Mouse [ChEMBL: CHEMBL3069] [UniProtKB: O35627]
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  • Constitutive androstane receptor in Mouse [GtoPdb: 607] [UniProtKB: Q3V008]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Constitutive androstane receptor in Mouse (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3069] [UniProtKB: O35627]
ChEMBL Inhibitory concentration against mammalian m-constitutive androstane receptor (mCAR) activity B 6.6 pIC50 250 nM IC50 J Med Chem (2003) 46: 4687-4695 [PMID:14561088]
Constitutive androstane receptor in Mouse [GtoPdb: 607] [UniProtKB: Q3V008]
GtoPdb - - 6.4 pIC50 - - - Nature (1998) 395: 612-5 [PMID:9783588]

ChEMBL data shown on this page come from version 32:

Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]