androstenol [Ligand Id: 2761] activity data from GtoPdb and ChEMBL

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

ChEMBL ligand: CHEMBL142348 (Androstenol)
  • Constitutive androstane receptor in Mouse [ChEMBL: CHEMBL3069] [UniProtKB: O35627]
There should be some charts here, you may need to enable JavaScript!
  • Constitutive androstane receptor in Mouse [GtoPdb: 607] [UniProtKB: Q3V008]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Constitutive androstane receptor in Mouse (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3069] [UniProtKB: O35627]
ChEMBL Inhibitory concentration against mammalian m-constitutive androstane receptor (mCAR) activity B 6.6 pIC50 250 nM IC50 J. Med. Chem. (2003) 46: 4687-4695 [PMID:14561088]
Constitutive androstane receptor in Mouse [GtoPdb: 607] [UniProtKB: Q3V008]
GtoPdb - - 6.4 pIC50 - - - Nature (1998) 395: 612-5 [PMID:9783588]

ChEMBL data shown on this page come from version 31:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]