androstenol [Ligand Id: 2761] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL142348 (Androstenol)
  • Constitutive androstane receptor in Mouse [ChEMBL: CHEMBL3069] [UniProtKB: O35627]
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  • Constitutive androstane receptor in Mouse [GtoPdb: 607] [UniProtKB: Q3V008]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Constitutive androstane receptor in Mouse (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3069] [UniProtKB: O35627]
ChEMBL Inhibitory concentration against mammalian m-constitutive androstane receptor (mCAR) activity B 6.6 pIC50 250 nM IC50 J. Med. Chem. (2003) 46: 4687-4695 [PMID:14561088]
Constitutive androstane receptor in Mouse [GtoPdb: 607] [UniProtKB: Q3V008]
GtoPdb - - 6.4 pIC50 - - - Nature (1998) 395: 612-5 [PMID:9783588]

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]