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ChEMBL ligand: CHEMBL142348 (Androstenol) |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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Constitutive androstane receptor in Mouse (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3069] [UniProtKB: O35627] | ||||||||
ChEMBL | Inhibitory concentration against mammalian m-constitutive androstane receptor (mCAR) activity | B | 6.6 | pIC50 | 250 | nM | IC50 | J. Med. Chem. (2003) 46: 4687-4695 [PMID:14561088] |
Constitutive androstane receptor in Mouse [GtoPdb: 607] [UniProtKB: Q3V008] | ||||||||
GtoPdb | - | - | 6.4 | pIC50 | - | - | - | Nature (1998) 395: 612-5 [PMID:9783588] |
ChEMBL data shown on this page come from version 31:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]