1-allyl-2-[3-(isopropylamino)propoxy]-9H-carbazole [Ligand Id: 3136] activity data from GtoPdb

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  • squalene synthase in Human [GtoPdb: 645] [UniProtKB: P37268]
  • squalene synthase in Rat [GtoPdb: 645] [UniProtKB: Q02769]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
squalene synthase in Human [GtoPdb: 645] [UniProtKB: P37268]
GtoPdb in vitro. Rat and human liver microsomes assayed using the Amin technique. - 7.49 pIC50 32 nM IC50 Bioorg. Med. Chem. (2004) 12: 5899-908 [PMID:15498666]
squalene synthase in Rat [GtoPdb: 645] [UniProtKB: Q02769]
GtoPdb in vitro. Rat and human liver microsomes assayed using the Amin technique. - 7.18 pIC50 66 nM IC50 Bioorg. Med. Chem. (2004) 12: 5899-908 [PMID:15498666]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.