guanylpirenzepine | Ligand Activity Charts | IUPHAR/BPS Guide to PHARMACOLOGY

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guanylpirenzepine
Ligand Activity Charts

guanylpirenzepine [Ligand Id: 3276] activity data from GtoPdb

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M₁ receptor in Rat [GtoPdb: 13] [UniProtKB: P08482] There should be some charts here, you may need to enable JavaScript!
M₂ receptor in Rat [GtoPdb: 14] [UniProtKB: P10980] There should be some charts here, you may need to enable JavaScript!
M₃ receptor in Rat [GtoPdb: 15] [UniProtKB: P08483] There should be some charts here, you may need to enable JavaScript!
M₄ receptor in Rat [GtoPdb: 16] [UniProtKB: P08485] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
M₁ receptor in Rat [GtoPdb: 13] [UniProtKB: P08482]
GtoPdb	-	-	7.6	pKi	-	-	-	Eur J Pharmacol (1996) 305: 187-92 [PMID:8813552]; Gen Pharmacol (1999) 32: 505-11 [PMID:10323493]
M₂ receptor in Rat [GtoPdb: 14] [UniProtKB: P10980]
GtoPdb	-	-	5.3	pKi	-	-	-	Eur J Pharmacol (1996) 305: 187-92 [PMID:8813552]
M₃ receptor in Rat [GtoPdb: 15] [UniProtKB: P08483]
GtoPdb	-	-	6.2	pKi	-	-	-	Eur J Pharmacol (1996) 305: 187-92 [PMID:8813552]
M₄ receptor in Rat [GtoPdb: 16] [UniProtKB: P08485]
GtoPdb	-	-	6.2	pKi	-	-	-	Eur J Pharmacol (1996) 305: 187-92 [PMID:8813552]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.