derenofylline [Ligand Id: 3281] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| A1 receptor in Human [GtoPdb: 18] [UniProtKB: P30542] | ||||||||
| GtoPdb | - | - | 9 | pKi | 1 | nM | Ki | Br J Pharmacol (2007) 151: 1025-32 [PMID:17558436] |
| A1 receptor in Rat [GtoPdb: 18] [UniProtKB: P25099] | ||||||||
| GtoPdb | - | - | 8.6 | pKi | 2.51 | nM | Ki | Br J Pharmacol (2007) 151: 1025-32 [PMID:17558436] |
| A2A receptor in Human [GtoPdb: 19] [UniProtKB: P29274] | ||||||||
| GtoPdb | - | - | 6.4 | pKi | 398 | nM | Ki | Br J Pharmacol (2007) 151: 1025-32 [PMID:17558436] |
| A2B receptor in Human [GtoPdb: 20] [UniProtKB: P29275] | ||||||||
| GtoPdb | - | - | 5.4 | pKi | 3981 | nM | Ki | Br J Pharmacol (2007) 151: 1025-32 [PMID:17558436] |
| A2B receptor in Rat [GtoPdb: 20] [UniProtKB: P29276] | ||||||||
| GtoPdb | - | - | 6.3 | pKi | 501 | nM | Ki | Br J Pharmacol (2007) 151: 1025-32 [PMID:17558436] |
| A3 receptor in Human [GtoPdb: 21] [UniProtKB: P0DMS8] | ||||||||
| GtoPdb | - | - | 6.7 | pKi | 200 | nM | Ki | Br J Pharmacol (2007) 151: 1025-32 [PMID:17558436] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
