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1
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secretin receptor
Rat
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2
_lig_chart_2
PAC1 receptor
Rat
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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secretin receptor in Rat [GtoPdb: 252] [UniProtKB: P23811] | ||||||||
GtoPdb | Inhibition of [125I]Tyr25 secretin binding in membranes from CHO cells expressing recombinant receptor | - | 7.7 | pIC50 | 20 | nM | IC50 | Peptides (1997) 18: 1539-45 [PMID:9437714] |
PAC1 receptor in Rat [GtoPdb: 370] [UniProtKB: P32215] | ||||||||
GtoPdb | Inhibition of [125I]-Ac-His1-PACAP-27 binding in membranes from CHO cells expressing recombinant receptor | - | 4.7 | pIC50 | 20000 | nM | IC50 | Peptides (1997) 18: 1539-45 [PMID:9437714] |
VPAC1 receptor in Human [GtoPdb: 371] [UniProtKB: P32241] | ||||||||
GtoPdb | Inhibition of [125I]VIP binding in membranes from LoVo cells expressing recombinant receptor | - | 7.2 | pIC50 | 60 | nM | IC50 | Peptides (1997) 18: 1539-45 [PMID:9437714] |
VPAC1 receptor in Rat [GtoPdb: 371] [UniProtKB: P30083] | ||||||||
GtoPdb | Inhibition of [125I]VIP binding in membranes from CHO cells expressing recombinant receptor | - | 9 | pIC50 | 1 | nM | IC50 | Peptides (1997) 18: 1539-45 [PMID:9437714] |
VPAC2 receptor in Human [GtoPdb: 372] [UniProtKB: P41587] | ||||||||
GtoPdb | Inhibition of [125I]VIP binding in membranes from CHO cells expressing recombinant receptor | - | 5.3 | pIC50 | 5000 | nM | IC50 | Peptides (1997) 18: 1539-45 [PMID:9437714] |
VPAC2 receptor in Rat [GtoPdb: 372] [UniProtKB: P35000] | ||||||||
GtoPdb | Inhibition of [125I]VIP binding in membranes from CHO cells expressing recombinant receptor | - | 5 | pIC50 | 10000 | nM | IC50 | Peptides (1997) 18: 1539-45 [PMID:9437714] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.