[Arg16]chicken secretin [Ligand Id: 3293] activity data from GtoPdb

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  • secretin receptor in Rat [GtoPdb: 252] [UniProtKB: P23811]
  • This target only has 0 pki data point
1 _lig_chart_1 secretin receptor Rat
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  • PAC1 receptor in Rat [GtoPdb: 370] [UniProtKB: P32215]
  • This target only has 0 pki data point
2 _lig_chart_2 PAC1 receptor Rat
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  • VPAC1 receptor in Human [GtoPdb: 371] [UniProtKB: P32241]
  • VPAC1 receptor in Rat [GtoPdb: 371] [UniProtKB: P30083]
  • This target only has 0 pki data point
3 _lig_chart_3 VPAC1 receptor HumanRat
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  • VPAC2 receptor in Human [GtoPdb: 372] [UniProtKB: P41587]
  • VPAC2 receptor in Rat [GtoPdb: 372] [UniProtKB: P35000]
  • This target only has 0 pki data point
4 _lig_chart_4 VPAC2 receptor HumanRat
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
secretin receptor in Rat [GtoPdb: 252] [UniProtKB: P23811]
GtoPdb Inhibition of [125I]Tyr25 secretin binding in membranes from CHO cells expressing recombinant receptor - 7.7 pIC50 20 nM IC50 Peptides (1997) 18: 1539-45 [PMID:9437714]
PAC1 receptor in Rat [GtoPdb: 370] [UniProtKB: P32215]
GtoPdb Inhibition of [125I]-Ac-His1-PACAP-27 binding in membranes from CHO cells expressing recombinant receptor - 4.7 pIC50 20000 nM IC50 Peptides (1997) 18: 1539-45 [PMID:9437714]
VPAC1 receptor in Human [GtoPdb: 371] [UniProtKB: P32241]
GtoPdb Inhibition of [125I]VIP binding in membranes from LoVo cells expressing recombinant receptor - 7.2 pIC50 60 nM IC50 Peptides (1997) 18: 1539-45 [PMID:9437714]
VPAC1 receptor in Rat [GtoPdb: 371] [UniProtKB: P30083]
GtoPdb Inhibition of [125I]VIP binding in membranes from CHO cells expressing recombinant receptor - 9 pIC50 1 nM IC50 Peptides (1997) 18: 1539-45 [PMID:9437714]
VPAC2 receptor in Human [GtoPdb: 372] [UniProtKB: P41587]
GtoPdb Inhibition of [125I]VIP binding in membranes from CHO cells expressing recombinant receptor - 5.3 pIC50 5000 nM IC50 Peptides (1997) 18: 1539-45 [PMID:9437714]
VPAC2 receptor in Rat [GtoPdb: 372] [UniProtKB: P35000]
GtoPdb Inhibition of [125I]VIP binding in membranes from CHO cells expressing recombinant receptor - 5 pIC50 10000 nM IC50 Peptides (1997) 18: 1539-45 [PMID:9437714]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.