M65 [Ligand Id: 3305] activity data from GtoPdb

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  • PAC1 receptor in Human [GtoPdb: 370] [UniProtKB: P41586]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
PAC1 receptor in Human [GtoPdb: 370] [UniProtKB: P41586]
GtoPdb inhibition of calcium influx stimulated by 30nM PACAP-27 in CHO cells stably expressing recombinant receptor - 6.6 pIC50 277.4 nM IC50 Neuropharmacology (2006) 51: 1086-98 [PMID:16930633]
GtoPdb inhibition of cyclic AMP formation stimulated by 0.1nM PACAP-27 in CHO cells stably expressing recombinant receptor - 6.8 pIC50 149.6 nM IC50 Neuropharmacology (2006) 51: 1086-98 [PMID:16930633]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.