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1
_lig_chart_1
M1 receptor
Human
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2
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M2 receptor
Human
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3
_lig_chart_3
M3 receptor
Human
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4
_lig_chart_4
M4 receptor
Human
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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M1 receptor in Human [GtoPdb: 13] [UniProtKB: P11229] | ||||||||
GtoPdb | - | - | 5 | pKd | - | - | - | Mol Pharmacol (1997) 52: 172-9 [PMID:9224827] |
M2 receptor in Human [GtoPdb: 14] [UniProtKB: P08172] | ||||||||
GtoPdb | - | - | 6.9 | pKd | - | - | - |
Mol Pharmacol (1997) 52: 172-9 [PMID:9224827]; Mol Pharmacol (2003) 64: 180-90 [PMID:12815174]; J Biol Chem (2007) 282: 25677-86 [PMID:17591774] |
M3 receptor in Human [GtoPdb: 15] [UniProtKB: P20309] | ||||||||
GtoPdb | - | - | 5.8 | pKd | - | - | - | Mol Pharmacol (1997) 52: 172-9 [PMID:9224827] |
M4 receptor in Human [GtoPdb: 16] [UniProtKB: P08173] | ||||||||
GtoPdb | - | - | 5.6 | pKd | - | - | - | Mol Pharmacol (1997) 52: 172-9 [PMID:9224827] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.