GSK Compound 34 [Ligand Id: 3502] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1082152
  • cyclin dependent kinase 19/Cell division cycle 2-like protein kinase 6 in Human [ChEMBL: CHEMBL6002] [GtoPdb: 1972] [UniProtKB: Q9BWU1]
  • This target only has 0 pki data point
1 CHEMBL1082152_lig_chart_1 Cell division cycle 2-like protein kinase 6 Human
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  • cyclin dependent kinase 8/Cell division protein kinase 8 in Human [ChEMBL: CHEMBL5719] [GtoPdb: 1980] [UniProtKB: P49336]
  • This target only has 0 pki data point
2 CHEMBL1082152_lig_chart_2 Cell division protein kinase 8 Human
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  • cyclin dependent kinase 2/Cyclin-dependent kinase 2 in Human [ChEMBL: CHEMBL301] [GtoPdb: 1973] [UniProtKB: P24941]
  • This target only has 0 pki data point
3 CHEMBL1082152_lig_chart_3 Cyclin-dependent kinase 2 Human
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  • cyclin dependent kinase 3/Cyclin-dependent kinase 3 in Human [ChEMBL: CHEMBL4442] [GtoPdb: 1975] [UniProtKB: Q00526]
  • This target only has 0 pki data point
4 CHEMBL1082152_lig_chart_4 Cyclin-dependent kinase 3 Human
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  • cyclin dependent kinase 5/Cyclin-dependent kinase 5 in Human [ChEMBL: CHEMBL4036] [GtoPdb: 1977] [UniProtKB: Q00535]
  • This target only has 0 pki data point
5 CHEMBL1082152_lig_chart_5 Cyclin-dependent kinase 5 Human
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  • cyclin dependent kinase 7/Cyclin-dependent kinase 7 in Human [ChEMBL: CHEMBL3055] [GtoPdb: 1979] [UniProtKB: P50613]
  • This target only has 0 pki data point
6 CHEMBL1082152_lig_chart_6 Cyclin-dependent kinase 7 Human
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  • cyclin dependent kinase 9/Cyclin-dependent kinase 9 in Human [ChEMBL: CHEMBL3116] [GtoPdb: 1981] [UniProtKB: P50750]
  • This target only has 0 pki data point
7 CHEMBL1082152_lig_chart_7 Cyclin-dependent kinase 9 Human
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  • CDC like kinase 2/Dual specificity protein kinase CLK2 in Human [ChEMBL: CHEMBL4225] [GtoPdb: 1991] [UniProtKB: P49760]
  • This target only has 0 pki data point
8 CHEMBL1082152_lig_chart_8 Dual specificity protein kinase CLK2 Human
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  • CDC like kinase 3/Dual specificity protein kinase CLK3 in Human [ChEMBL: CHEMBL4226] [GtoPdb: 1992] [UniProtKB: P49761]
  • This target only has 0 pki data point
9 CHEMBL1082152_lig_chart_9 Dual specificity protein kinase CLK3 Human
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  • CDC like kinase 4/Dual specificity protein kinase CLK4 in Human [ChEMBL: CHEMBL4203] [GtoPdb: 1993] [UniProtKB: Q9HAZ1]
  • This target only has 0 pki data point
10 CHEMBL1082152_lig_chart_10 Dual specificity protein kinase CLK4 Human
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  • TTK protein kinase/Dual specificity protein kinase TTK in Human [ChEMBL: CHEMBL3983] [GtoPdb: 2264] [UniProtKB: P33981]
  • This target only has 0 pki data point
11 CHEMBL1082152_lig_chart_11 Dual specificity protein kinase TTK Human
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  • dual specificity tyrosine phosphorylation regulated kinase 1B/Dual specificity tyrosine-phosphorylation-regulated kinase 1B in Human [ChEMBL: CHEMBL5543] [GtoPdb: 2010] [UniProtKB: Q9Y463]
  • This target only has 0 pki data point
12 CHEMBL1082152_lig_chart_12 Dual specificity tyrosine-phosphorylation-regulated kinase 1B Human
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  • CDC like kinase 1/Dual specificty protein kinase CLK1 in Human [ChEMBL: CHEMBL4224] [GtoPdb: 1990] [UniProtKB: P49759]
  • This target only has 0 pki data point
13 CHEMBL1082152_lig_chart_13 Dual specificty protein kinase CLK1 Human
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  • glycogen synthase kinase 3 alpha/Glycogen synthase kinase-3 alpha in Human [ChEMBL: CHEMBL2850] [GtoPdb: 2029] [UniProtKB: P49840]
  • This target only has 0 pki data point
14 CHEMBL1082152_lig_chart_14 Glycogen synthase kinase-3 alpha Human
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  • glycogen synthase kinase 3 beta/Glycogen synthase kinase-3 beta in Human [ChEMBL: CHEMBL262] [GtoPdb: 2030] [UniProtKB: P49841]
  • This target only has 0 pki data point
15 CHEMBL1082152_lig_chart_15 Glycogen synthase kinase-3 beta Human
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  • eukaryotic translation initiation factor 2 alpha kinase 2/Interferon-induced, double-stranded RNA-activated protein kinase in Human [ChEMBL: CHEMBL5785] [GtoPdb: 2016] [UniProtKB: P19525]
  • This target only has 0 pki data point
16 CHEMBL1082152_lig_chart_16 Interferon-induced, double-stranded RNA-activated protein kinase Human
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  • mitogen-activated protein kinase 3/MAP kinase ERK1 in Human [ChEMBL: CHEMBL3385] [GtoPdb: 1494] [UniProtKB: P27361]
  • This target only has 0 pki data point
17 CHEMBL1082152_lig_chart_17 MAP kinase ERK1 Human
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  • mitogen-activated protein kinase 1/MAP kinase ERK2 in Human [ChEMBL: CHEMBL4040] [GtoPdb: 1495] [UniProtKB: P28482]
  • This target only has 0 pki data point
18 CHEMBL1082152_lig_chart_18 MAP kinase ERK2 Human
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  • mitogen-activated protein kinase 15/Mitogen-activated protein kinase 15 in Human [ChEMBL: CHEMBL5198] [GtoPdb: 2090] [UniProtKB: Q8TD08]
  • This target only has 0 pki data point
19 CHEMBL1082152_lig_chart_19 Mitogen-activated protein kinase 15 Human
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  • mitogen-activated protein kinase 4/Mitogen-activated protein kinase 4 in Human [ChEMBL: CHEMBL5759] [GtoPdb: 2091] [UniProtKB: P31152]
  • This target only has 0 pki data point
20 CHEMBL1082152_lig_chart_20 Mitogen-activated protein kinase 4 Human
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  • mitogen-activated protein kinase 6/Mitogen-activated protein kinase 6 in Human [ChEMBL: CHEMBL5121] [GtoPdb: 2092] [UniProtKB: Q16659]
  • This target only has 0 pki data point
21 CHEMBL1082152_lig_chart_21 Mitogen-activated protein kinase 6 Human
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  • mitogen-activated protein kinase 7/Mitogen-activated protein kinase 7 in Human [ChEMBL: CHEMBL5332] [GtoPdb: 2093] [UniProtKB: Q13164]
  • This target only has 0 pki data point
22 CHEMBL1082152_lig_chart_22 Mitogen-activated protein kinase 7 Human
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  • protein kinase C alpha/Protein kinase C alpha in Human [ChEMBL: CHEMBL299] [GtoPdb: 1482] [UniProtKB: P17252]
  • This target only has 0 pki data point
23 CHEMBL1082152_lig_chart_23 Protein kinase C alpha Human
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  • serine/threonine kinase 16/Serine/threonine-protein kinase 16 in Human [ChEMBL: CHEMBL3938] [GtoPdb: 2213] [UniProtKB: O75716]
  • This target only has 0 pki data point
24 CHEMBL1082152_lig_chart_24 Serine/threonine-protein kinase 16 Human
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  • aurora kinase A/Serine/threonine-protein kinase Aurora-A in Human [ChEMBL: CHEMBL4722] [GtoPdb: 1936] [UniProtKB: O14965]
  • This target only has 0 pki data point
25 CHEMBL1082152_lig_chart_25 Serine/threonine-protein kinase Aurora-A Human
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  • aurora kinase B/Serine/threonine-protein kinase Aurora-B in Human [ChEMBL: CHEMBL2185] [GtoPdb: 1937] [UniProtKB: Q96GD4]
  • This target only has 0 pki data point
26 CHEMBL1082152_lig_chart_26 Serine/threonine-protein kinase Aurora-B Human
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  • aurora kinase C/Serine/threonine-protein kinase Aurora-C in Human [ChEMBL: CHEMBL3935] [GtoPdb: 1938] [UniProtKB: Q9UQB9]
  • This target only has 0 pki data point
27 CHEMBL1082152_lig_chart_27 Serine/threonine-protein kinase Aurora-C Human
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  • cyclin dependent kinase 16/Serine/threonine-protein kinase PCTAIRE-1 in Human [ChEMBL: CHEMBL4597] [GtoPdb: 1969] [UniProtKB: Q00536]
  • This target only has 0 pki data point
28 CHEMBL1082152_lig_chart_28 Serine/threonine-protein kinase PCTAIRE-1 Human
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  • cyclin dependent kinase 17/Serine/threonine-protein kinase PCTAIRE-2 in Human [ChEMBL: CHEMBL5790] [GtoPdb: 1970] [UniProtKB: Q00537]
  • This target only has 0 pki data point
29 CHEMBL1082152_lig_chart_29 Serine/threonine-protein kinase PCTAIRE-2 Human
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  • cyclin dependent kinase 18/Serine/threonine-protein kinase PCTAIRE-3 in Human [ChEMBL: CHEMBL5316] [GtoPdb: 1971] [UniProtKB: Q07002]
  • This target only has 0 pki data point
30 CHEMBL1082152_lig_chart_30 Serine/threonine-protein kinase PCTAIRE-3 Human
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  • polo like kinase 1/Serine/threonine-protein kinase PLK1 in Human [ChEMBL: CHEMBL3024] [GtoPdb: 2168] [UniProtKB: P53350]
  • This target only has 0 pki data point
31 CHEMBL1082152_lig_chart_31 Serine/threonine-protein kinase PLK1 Human
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  • polo like kinase 3/Serine/threonine-protein kinase PLK3 in Human [ChEMBL: CHEMBL4897] [GtoPdb: 2170] [UniProtKB: Q9H4B4]
  • This target only has 0 pki data point
32 CHEMBL1082152_lig_chart_32 Serine/threonine-protein kinase PLK3 Human
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  • polo like kinase 4/Serine/threonine-protein kinase PLK4 in Human [ChEMBL: CHEMBL3788] [GtoPdb: 2171] [UniProtKB: O00444]
  • This target only has 0 pki data point
33 CHEMBL1082152_lig_chart_33 Serine/threonine-protein kinase PLK4 Human
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  • CCR2 in Human [GtoPdb: 59] [UniProtKB: P41597]
  • This target only has 1 pki data point
34 CHEMBL1082152_lig_chart_34 CCR2 Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
cyclin dependent kinase 19/Cell division cycle 2-like protein kinase 6 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL6002] [GtoPdb: 1972] [UniProtKB: Q9BWU1]
ChEMBL Inhibition of CDK11 B 4.4 pKd 40000 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
cyclin dependent kinase 8/Cell division protein kinase 8 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5719] [GtoPdb: 1980] [UniProtKB: P49336]
ChEMBL Inhibition of CDK8 B 4.4 pKd 40000 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
cyclin dependent kinase 2/Cyclin-dependent kinase 2 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL301] [GtoPdb: 1973] [UniProtKB: P24941]
ChEMBL Inhibition of CDK2 B 6.82 pKd 150 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
cyclin dependent kinase 3/Cyclin-dependent kinase 3 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4442] [GtoPdb: 1975] [UniProtKB: Q00526]
ChEMBL Inhibition of CDK3 B 7.1 pKd 80 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
cyclin dependent kinase 5/Cyclin-dependent kinase 5 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4036] [GtoPdb: 1977] [UniProtKB: Q00535]
ChEMBL Inhibition of CDK5 B 5.17 pKd 6800 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
cyclin dependent kinase 7/Cyclin-dependent kinase 7 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3055] [GtoPdb: 1979] [UniProtKB: P50613]
ChEMBL Inhibition of CDK7 B 7.39 pKd 41 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
cyclin dependent kinase 9/Cyclin-dependent kinase 9 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3116] [GtoPdb: 1981] [UniProtKB: P50750]
ChEMBL Inhibition of CDK9 B 6.39 pKd 410 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
CDC like kinase 2/Dual specificity protein kinase CLK2 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4225] [GtoPdb: 1991] [UniProtKB: P49760]
ChEMBL Inhibition of CLK2 B 8 pKd 10 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
CDC like kinase 3/Dual specificity protein kinase CLK3 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4226] [GtoPdb: 1992] [UniProtKB: P49761]
ChEMBL Inhibition of CLK3 B 6.51 pKd 310 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
CDC like kinase 4/Dual specificity protein kinase CLK4 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4203] [GtoPdb: 1993] [UniProtKB: Q9HAZ1]
ChEMBL Inhibition of CLK4 B 6.96 pKd 110 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
TTK protein kinase/Dual specificity protein kinase TTK in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3983] [GtoPdb: 2264] [UniProtKB: P33981]
ChEMBL Inhibition of TTK B 5.17 pKd 6700 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
dual specificity tyrosine phosphorylation regulated kinase 1B/Dual specificity tyrosine-phosphorylation-regulated kinase 1B in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5543] [GtoPdb: 2010] [UniProtKB: Q9Y463]
ChEMBL Inhibition of DYRK1B B 7.06 pKd 87 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
CDC like kinase 1/Dual specificty protein kinase CLK1 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4224] [GtoPdb: 1990] [UniProtKB: P49759]
ChEMBL Inhibition of CLK1 B 7.8 pKd 16 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
glycogen synthase kinase 3 alpha/Glycogen synthase kinase-3 alpha in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2850] [GtoPdb: 2029] [UniProtKB: P49840]
ChEMBL Inhibition of GSK3alpha B 8.82 pKd 1.5 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
glycogen synthase kinase 3 beta/Glycogen synthase kinase-3 beta in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL262] [GtoPdb: 2030] [UniProtKB: P49841]
ChEMBL Inhibition of human recombinant GSK3-beta assessed as [gamma33]ATP transfer to biotinylated CREB-peptide substrate after 1 hr by scintillation counting B 10.28 pKd 0.05 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
ChEMBL Inhibition of human recombinant GSK3-beta assessed as [gamma33]ATP transfer to biotinylated CREB-peptide substrate after 1 hr by scintillation counting B 9.22 pIC50 0.6 nM IC50 Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
eukaryotic translation initiation factor 2 alpha kinase 2/Interferon-induced, double-stranded RNA-activated protein kinase in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5785] [GtoPdb: 2016] [UniProtKB: P19525]
ChEMBL Inhibition of PRKR B 4.85 pKd 14000 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
mitogen-activated protein kinase 3/MAP kinase ERK1 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3385] [GtoPdb: 1494] [UniProtKB: P27361]
ChEMBL Inhibition of ERK1 B 4.4 pKd 40000 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
mitogen-activated protein kinase 1/MAP kinase ERK2 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4040] [GtoPdb: 1495] [UniProtKB: P28482]
ChEMBL Inhibition of ERK2 B 4.4 pKd 40000 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
mitogen-activated protein kinase 15/Mitogen-activated protein kinase 15 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5198] [GtoPdb: 2090] [UniProtKB: Q8TD08]
ChEMBL Inhibition of ERK8 B 7.49 pKd 32 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
mitogen-activated protein kinase 4/Mitogen-activated protein kinase 4 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5759] [GtoPdb: 2091] [UniProtKB: P31152]
ChEMBL Inhibition of ERK4 B 4.4 pKd 40000 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
mitogen-activated protein kinase 6/Mitogen-activated protein kinase 6 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5121] [GtoPdb: 2092] [UniProtKB: Q16659]
ChEMBL Inhibition of ERK3 B 4.4 pKd 40000 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
mitogen-activated protein kinase 7/Mitogen-activated protein kinase 7 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5332] [GtoPdb: 2093] [UniProtKB: Q13164]
ChEMBL Inhibition of ERK5 B 5.25 pKd 5600 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
protein kinase C alpha/Protein kinase C alpha in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL299] [GtoPdb: 1482] [UniProtKB: P17252]
ChEMBL Inhibition of PKCalpha B 6.4 pIC50 400 nM IC50 Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
serine/threonine kinase 16/Serine/threonine-protein kinase 16 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3938] [GtoPdb: 2213] [UniProtKB: O75716]
ChEMBL Inhibition of STK16 B 6.64 pKd 230 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
aurora kinase A/Serine/threonine-protein kinase Aurora-A in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4722] [GtoPdb: 1936] [UniProtKB: O14965]
ChEMBL Inhibition of AURKA B 4.4 pKd 40000 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
aurora kinase B/Serine/threonine-protein kinase Aurora-B in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2185] [GtoPdb: 1937] [UniProtKB: Q96GD4]
ChEMBL Inhibition of AURKB B 4.4 pKd 40000 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
aurora kinase C/Serine/threonine-protein kinase Aurora-C in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3935] [GtoPdb: 1938] [UniProtKB: Q9UQB9]
ChEMBL Inhibition of AURKC B 4.64 pKd 23000 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
cyclin dependent kinase 16/Serine/threonine-protein kinase PCTAIRE-1 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4597] [GtoPdb: 1969] [UniProtKB: Q00536]
ChEMBL Inhibition of PCTK1 B 7.92 pKd 12 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
cyclin dependent kinase 17/Serine/threonine-protein kinase PCTAIRE-2 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5790] [GtoPdb: 1970] [UniProtKB: Q00537]
ChEMBL Inhibition of PCTK2 B 7.16 pKd 69 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
cyclin dependent kinase 18/Serine/threonine-protein kinase PCTAIRE-3 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5316] [GtoPdb: 1971] [UniProtKB: Q07002]
ChEMBL Inhibition of PCTK3 B 6.96 pKd 110 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
polo like kinase 1/Serine/threonine-protein kinase PLK1 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3024] [GtoPdb: 2168] [UniProtKB: P53350]
ChEMBL Inhibition of PLK1 B 4.64 pKd 23000 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
polo like kinase 3/Serine/threonine-protein kinase PLK3 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4897] [GtoPdb: 2170] [UniProtKB: Q9H4B4]
ChEMBL Inhibition of PLK3 B 4.4 pKd 40000 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
polo like kinase 4/Serine/threonine-protein kinase PLK4 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3788] [GtoPdb: 2171] [UniProtKB: O00444]
ChEMBL Inhibition of PLK4 B 6.49 pKd 320 nM Kd Bioorg. Med. Chem. Lett. (2010) 20: 1693-1696 [PMID:20138512]
CCR2 in Human [GtoPdb: 59] [UniProtKB: P41597]
GtoPdb - - 7.6 pKi 25.1 nM Ki

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]