galanin [Ligand Id: 3592] activity data from GtoPdb

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  • GAL1 receptor in Human [GtoPdb: 243] [UniProtKB: P47211]
  • GAL1 receptor in Rat [GtoPdb: 243] [UniProtKB: Q62805]
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  • GAL2 receptor in Human [GtoPdb: 244] [UniProtKB: O43603]
  • GAL2 receptor in Rat [GtoPdb: 244] [UniProtKB: O08726]
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  • GAL3 receptor in Human [GtoPdb: 245] [UniProtKB: O60755]
  • GAL3 receptor in Rat [GtoPdb: 245] [UniProtKB: O88626]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
GAL1 receptor in Human [GtoPdb: 243] [UniProtKB: P47211]
GtoPdb - - 10.51 pKi 0.03 nM Ki J Pharmacol Exp Ther (1998) 287: 448-56 [PMID:9808667];
Peptides (1998) 19: 1771-81 [PMID:9880084];
Proc Natl Acad Sci USA (1994) 91: 9780-3 [PMID:7524088];
Regul Pept (2001) 102: 15-9 [PMID:11600206]
GtoPdb - - 9.89 pIC50 0.13 nM IC50 Proc Natl Acad Sci USA (2001) 98: 9960-4 [PMID:11481429];
Biochem Biophys Res Commun (1997) 233: 823-8 [PMID:9168941];
Brain Res Mol Brain Res (1998) 58: 156-69 [PMID:9685625]
GAL1 receptor in Rat [GtoPdb: 243] [UniProtKB: Q62805]
GtoPdb - - 9.85 pKi 0.14 nM Ki J Biol Chem (1998) 273: 23321-6 [PMID:9722565];
J Mol Neurosci (1995) 6: 33-41 [PMID:8562318]
GtoPdb - - 10.22 pIC50 0.06 nM IC50 Biochem Biophys Res Commun (1997) 233: 823-8 [PMID:9168941];
FEBS Lett (1997) 405: 285-90 [PMID:9108306]
GAL2 receptor in Human [GtoPdb: 244] [UniProtKB: O43603]
GtoPdb - - 9.07 pKi 0.86 nM Ki Peptides (1998) 19: 1771-81 [PMID:9880084];
Regul Pept (2001) 102: 15-9 [PMID:11600206];
Biochem Biophys Res Commun (1998) 243: 474-9 [PMID:9480833]
GtoPdb - - 9.29 pIC50 0.51 nM IC50 Brain Res Mol Brain Res (1998) 58: 156-69 [PMID:9685625]
GtoPdb - - 9.15 pEC50 0.71 nM EC50 Peptides (1998) 19: 1771-81 [PMID:9880084];
Brain Res Mol Brain Res (1998) 58: 156-69 [PMID:9685625]
GAL2 receptor in Rat [GtoPdb: 244] [UniProtKB: O08726]
GtoPdb - - 8.6 pKi 2.51 nM Ki J Biol Chem (1998) 273: 23321-6 [PMID:9722565]
GtoPdb - - 9 pIC50 1 nM IC50 Brain Res Mol Brain Res (1997) 51: 49-59 [PMID:9427506];
Proc Natl Acad Sci USA (2001) 98: 9960-4 [PMID:11481429];
FEBS Lett (1997) 405: 285-90 [PMID:9108306]
GAL3 receptor in Human [GtoPdb: 245] [UniProtKB: O60755]
GtoPdb - - 7.16 pKi 69.18 nM Ki J Biol Chem (1998) 273: 23321-6 [PMID:9722565];
Peptides (1998) 19: 1771-81 [PMID:9880084]
GtoPdb - - 7.12 pIC50 75 nM IC50 J Neurochem (1998) 71: 2239-51 [PMID:9832121]
GAL3 receptor in Rat [GtoPdb: 245] [UniProtKB: O88626]
GtoPdb - - 7.28 pKi 52.48 nM Ki J Biol Chem (1998) 273: 23321-6 [PMID:9722565]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.