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ChEMBL ligand: CHEMBL2110824 (Buserelin, Suprecur, Suprefact) |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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GnRH1 receptor in Human [GtoPdb: 256] [UniProtKB: P30968] | ||||||||
GtoPdb | - | - | 10.4 | pKd | 0.04 | nM | Kd |
Br J Pharmacol (2016) 173: 128-41 [PMID:26398856]; Biosens Bioelectron (2016) 79: 721-7 [PMID:26774084] |
GtoPdb | - | - | 10 | pKi | 0.1 | nM | Ki | Br J Pharmacol (2016) 173: 128-41 [PMID:26398856] |
GtoPdb | - | - | 10.52 | pEC50 | 0.03 | nM | EC50 | Biosens Bioelectron (2016) 79: 721-7 [PMID:26774084] |
GnRH1 receptor in Mouse [GtoPdb: 256] [UniProtKB: Q01776] | ||||||||
GtoPdb | - | - | 10.05 | pEC50 | 0.09 | nM | EC50 | Biosens Bioelectron (2016) 79: 721-7 [PMID:26774084] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]