C7 [Ligand Id: 3861] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| GAL1 receptor in Human [GtoPdb: 243] [UniProtKB: P47211] | ||||||||
| GtoPdb | - | - | 10.09 | pKi | 0.08 | nM | Ki |
J Pharmacol Exp Ther (1998) 287: 448-56 [PMID:9808667]; Peptides (1998) 19: 1771-81 [PMID:9880084] |
| GtoPdb | - | - | 8.98 | pIC50 | 1.04 | nM | IC50 |
Biochem Biophys Res Commun (1997) 233: 823-8 [PMID:9168941]; Brain Res Mol Brain Res (1998) 58: 156-69 [PMID:9685625] |
| GAL1 receptor in Mouse [GtoPdb: 243] [UniProtKB: P56479] | ||||||||
| GtoPdb | - | - | 9.02 | pKi | 0.96 | nM | Ki |
FEBS Lett (1997) 411: 225-30 [PMID:9271210]; J Neurochem (1998) 71: 2252-9 [PMID:9832122] |
| GAL1 receptor in Rat [GtoPdb: 243] [UniProtKB: Q62805] | ||||||||
| GtoPdb | - | - | 9.55 | pKi | 0.28 | nM | Ki |
J Biol Chem (1997) 272: 24612-6 [PMID:9305929]; J Biol Chem (1998) 273: 23321-6 [PMID:9722565]; Brain Res Mol Brain Res (1995) 34: 179-89 [PMID:8750821] |
| GtoPdb | - | - | 8.31 | pIC50 | 4.9 | nM | IC50 |
Biochem Biophys Res Commun (1997) 233: 823-8 [PMID:9168941]; FEBS Lett (1997) 405: 285-90 [PMID:9108306] |
| GAL2 receptor in Human [GtoPdb: 244] [UniProtKB: O43603] | ||||||||
| GtoPdb | - | - | 9.2 | pKi | 0.63 | nM | Ki |
Peptides (1998) 19: 1771-81 [PMID:9880084]; Biochem Biophys Res Commun (1998) 243: 474-9 [PMID:9480833] |
| GtoPdb | - | - | 8.08 | pIC50 | 8.39 | nM | IC50 | Brain Res Mol Brain Res (1998) 58: 156-69 [PMID:9685625] |
| GtoPdb | - | - | 8.03 | pEC50 | 9.33 | nM | EC50 | Peptides (1998) 19: 1771-81 [PMID:9880084] |
| GAL2 receptor in Mouse [GtoPdb: 244] [UniProtKB: O88854] | ||||||||
| GtoPdb | - | - | 7.85 | pKi | 14 | nM | Ki | J Neurochem (1998) 71: 2252-9 [PMID:9832122] |
| GAL2 receptor in Rat [GtoPdb: 244] [UniProtKB: O08726] | ||||||||
| GtoPdb | - | - | 9.25 | pKi | 0.56 | nM | Ki |
J Biol Chem (1997) 272: 24612-6 [PMID:9305929]; J Biol Chem (1998) 273: 23321-6 [PMID:9722565]; Mol Pharmacol (1997) 52: 337-43 [PMID:9281594]; J Neurochem (1998) 71: 2252-9 [PMID:9832122] |
| GtoPdb | - | - | 8.44 | pIC50 | 3.6 | nM | IC50 |
Brain Res Mol Brain Res (1997) 51: 49-59 [PMID:9427506]; FEBS Lett (1997) 405: 285-90 [PMID:9108306] |
| GtoPdb | - | - | 8.52 | pEC50 | 3 | nM | EC50 | J Biol Chem (1997) 272: 24612-6 [PMID:9305929] |
| GAL3 receptor in Human [GtoPdb: 245] [UniProtKB: O60755] | ||||||||
| GtoPdb | - | - | 8.08 | pKi | 8.31 | nM | Ki |
J Biol Chem (1998) 273: 23321-6 [PMID:9722565]; Peptides (1998) 19: 1771-81 [PMID:9880084] |
| GAL3 receptor in Rat [GtoPdb: 245] [UniProtKB: O88626] | ||||||||
| GtoPdb | - | - | 9.12 | pKi | 0.75 | nM | Ki |
J Biol Chem (1998) 273: 23321-6 [PMID:9722565]; J Biol Chem (1997) 272: 31949-52 [PMID:9405385] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
