M35 [Ligand Id: 3898] activity data from GtoPdb

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  • GAL1 receptor in Human [GtoPdb: 243] [UniProtKB: P47211]
  • GAL1 receptor in Rat [GtoPdb: 243] [UniProtKB: Q62805]
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  • GAL2 receptor in Human [GtoPdb: 244] [UniProtKB: O43603]
  • GAL2 receptor in Mouse [GtoPdb: 244] [UniProtKB: O88854]
  • GAL2 receptor in Rat [GtoPdb: 244] [UniProtKB: O08726]
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  • GAL3 receptor in Human [GtoPdb: 245] [UniProtKB: O60755]
  • GAL3 receptor in Rat [GtoPdb: 245] [UniProtKB: O88626]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
GAL1 receptor in Human [GtoPdb: 243] [UniProtKB: P47211]
GtoPdb - - 10.92 pKi 0.01 nM Ki J. Pharmacol. Exp. Ther. (1998) 287: 448-56 [PMID:9808667];
Peptides (1998) 19: 1771-81 [PMID:9880084];
Neuropeptides (2005) 39: 143-6 [PMID:15944002]
GtoPdb - - 10.4 pIC50 0.04 nM IC50 Biochem. Biophys. Res. Commun. (1997) 233: 823-8 [PMID:9168941]
GAL1 receptor in Rat [GtoPdb: 243] [UniProtKB: Q62805]
GtoPdb - - 9.52 pKi 0.3 nM Ki J. Biol. Chem. (1997) 272: 24612-6 [PMID:9305929];
J. Biol. Chem. (1998) 273: 23321-6 [PMID:9722565];
Brain Res. Mol. Brain Res. (1995) 34: 179-89 [PMID:8750821]
GtoPdb - - 11 pIC50 0.01 nM IC50 Biochem. Biophys. Res. Commun. (1997) 233: 823-8 [PMID:9168941];
FEBS Lett. (1997) 405: 285-90 [PMID:9108306]
GAL2 receptor in Human [GtoPdb: 244] [UniProtKB: O43603]
GtoPdb - - 8.74 pKi 1.8 nM Ki Peptides (1998) 19: 1771-81 [PMID:9880084];
Biochem. Biophys. Res. Commun. (1998) 243: 474-9 [PMID:9480833]
GtoPdb - - 9.14 pEC50 0.72 nM EC50 Peptides (1998) 19: 1771-81 [PMID:9880084];
Brain Res. Mol. Brain Res. (1998) 58: 156-69 [PMID:9685625]
GAL2 receptor in Mouse [GtoPdb: 244] [UniProtKB: O88854]
GtoPdb - - 8.31 pKi 4.9 nM Ki J. Neurochem. (1998) 71: 2252-9 [PMID:9832122]
GAL2 receptor in Rat [GtoPdb: 244] [UniProtKB: O08726]
GtoPdb - - 9.22 pKi 0.6 nM Ki J. Biol. Chem. (1997) 272: 24612-6 [PMID:9305929];
J. Biol. Chem. (1998) 273: 23321-6 [PMID:9722565];
Mol. Pharmacol. (1997) 52: 337-43 [PMID:9281594];
J. Neurochem. (1998) 71: 2252-9 [PMID:9832122];
Neuropeptides (2005) 39: 143-6 [PMID:15944002]
GtoPdb - - 9.37 pIC50 0.43 nM IC50 Brain Res. Mol. Brain Res. (1997) 51: 49-59 [PMID:9427506];
FEBS Lett. (1997) 405: 285-90 [PMID:9108306]
GtoPdb - - 7.54 pEC50 29 nM EC50 J. Biol. Chem. (1997) 272: 24612-6 [PMID:9305929]
GAL3 receptor in Human [GtoPdb: 245] [UniProtKB: O60755]
GtoPdb - - 7.84 pKi 14.45 nM Ki J. Biol. Chem. (1998) 273: 23321-6 [PMID:9722565];
Peptides (1998) 19: 1771-81 [PMID:9880084];
International Journal of Peptide Research and Therapeutics (2010) : 17-22
GAL3 receptor in Rat [GtoPdb: 245] [UniProtKB: O88626]
GtoPdb - - 8.68 pKi 2.09 nM Ki J. Biol. Chem. (1998) 273: 23321-6 [PMID:9722565];
J. Biol. Chem. (1997) 272: 31949-52 [PMID:9405385];
Neuropeptides (2005) 39: 143-6 [PMID:15944002]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.