[3H]cytisine [Ligand Id: 3979] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1628606
  • nicotinic acetylcholine receptor α4 subunit in Human [GtoPdb: 465] [UniProtKB: P43681]
  • nicotinic acetylcholine receptor α4 subunit in Rat [GtoPdb: 465] [UniProtKB: P09483]
  • This target only has 0 pki data point
  • 0
1 CHEMBL1628606_lig_chart_1 nicotinic acetylcholine receptor α4 subunit HumanRat
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
nicotinic acetylcholine receptor α4 subunit in Human [GtoPdb: 465] [UniProtKB: P43681]
GtoPdb - - 9.37 pKd 0.43 nM Kd
GtoPdb - - 10 pKd 0.1 nM Kd
nicotinic acetylcholine receptor α4 subunit in Rat [GtoPdb: 465] [UniProtKB: P09483]
GtoPdb - - 10 pKd 0.1 nM Kd

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]