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ChEMBL ligand: CHEMBL1232313 (Domoic Acid) |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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GluK2 in Human [GtoPdb: 451] [UniProtKB: Q13002] | ||||||||
GtoPdb | Measuring displacement of [3H]Kainate binding by domoate. | - | 7.74 | pKi | 18.3 | nM | Ki | J Med Chem (1996) 39: 3617-24 [PMID:8809152] |
GluK3 in Rat [GtoPdb: 452] [UniProtKB: P42264] | ||||||||
GtoPdb | - | - | 8.42 | pKi | 3.84 | nM | Ki | J Med Chem (2008) 51: 4093-103 [PMID:18578478] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]