kainate [Ligand Id: 4231] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| GluK1 in Human [GtoPdb: 450] [UniProtKB: P39086] | ||||||||
| GtoPdb | - | - | 6.75 | pKi | 177 | nM | Ki | Neuropharmacology (1998) 37: 1261-7 [PMID:9849663] |
| GluK2 in Human [GtoPdb: 451] [UniProtKB: Q13002] | ||||||||
| GtoPdb | Measured using kainic acid. | - | 7.49 | pKi | 32 | nM | Ki |
J Med Chem (1996) 39: 3617-24 [PMID:8809152]; Neuropharmacology (1998) 37: 1261-7 [PMID:9849663] |
| GluK2 in Rat [GtoPdb: 451] [UniProtKB: P42260] | ||||||||
| GtoPdb | Measured using kainic acid in rat forebrain homogenate. | - | 8.43 | pKi | 3.7 | nM | Ki |
J Pharmacol Exp Ther (1997) 280: 422-7 [PMID:8996224]; J Med Chem (1996) 39: 3617-24 [PMID:8809152] |
| GluK3 in Rat [GtoPdb: 452] [UniProtKB: P42264] | ||||||||
| GtoPdb | - | - | 7.48 | pKi | 32.8 | nM | Ki | J Med Chem (2008) 51: 4093-103 [PMID:18578478] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
